产品名称

BIA 10-2474

一般描述

BIA10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH).

别 称

N-cyclohexyl-N-methyl-4-(1-oxidopyridin-1-ium-3-yl)imidazole-1-carboxamide;BIA-10-2474; BIA10-2474

纯 度

≥98.5%(HPLC)

CAS NO.

1233855-46-3

分子式

C¹⁶H²⁰N⁴O²

分子量

300.36

适用范围

生物试剂，适用于细胞培养等

l  理化信息

外 观

白色或类白色固体

l  生物学信息

生物活性/药理作用

BIA10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central nervous system and in peripheral tissues (that is, the rest of the body other than the brain and spinal cord). BIA 10-2474 interacts with the human endocannabinoid system. BIA 10-2474 was in development for the treatment of a range of different medical conditions from anxiety to Parkinson's disease,   also for the treatment of chronic pain of multiple sclerosis, Y, hypertension or the treatment of obesity.

l  包装与存储

包 装

5mg; 10mg

存储温度

-20℃

l  注意事项及免责声明

本产品仅用于实验研究，不得作为药物使用，不得用于家用或其它用途。

l  参考文献

1.    http://www.drugbank.ca

2.    https://ncit.nci.nih.gov

3.    https://www.ncbi.nlm.nih.gov