产品名称

Cyclobenzaprine HCl(盐酸环苯扎林)

一般描述

Cyclobenzaprine HCl is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms A 5-HT2 receptor antagonist.   

别 称

N,N-dimethyl-3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propan-1-amine; hydrochloride

纯 度

≥98.0%(HPLC)

CAS NO.

6202-23-9

分子式

C²⁰H²²ClN

分子量

311.853

适用范围

生物试剂，适用于细胞培养等

l  理化信息

外 观

固体

溶解性(25°C)

DMSO

≥50mg/ml

水

≥50mg/ml

l  生物学信息

生物活性/药理作用

Cyclobenzaprine Hydrochloride is a centrally acting muscle relaxant, chemically similar to amitriptyline hydrochloride with antidepressant activity. The exact mechanism of action of cyclobenzaprine hydrochloride has not been fully determined. However, it primarily acts at the brain stem to reduce tonic somatic motor activity, influencing both gamma and alpha motor   neurons. This leads to a reduction in muscle spasms.

应 用

1.Muscle Relaxants, Central

2.Tranquilizing Agents

3.Antidepressive Agents, Tricyclic

l  存储

存储温度

-20°C

l  注意事项及免责声明

本产品仅用于实验研究，不得作为药物使用，不得用于家用或其它用途。

l  参考文献

1.    http://www.drugbank.ca

2.    https://ncit.nci.nih.gov

3.  https://www.ncbi.nlm.nih.gov