EPZ004777 is a potent, selective DOT1L inhibitor.

AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor.

GSK J4 HCl is a cell permeable prodrug of GSK J1.

JIB-04 is a pan-selective Jumonji histone demethylase inhibitor.

ORY-1001 2HCl is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor.

(+)-JQ1 is a BET bromodomain inhibitor.

I-BET151 is a novel selective BET inhibitor.

Molibresib is an inhibitor for BET proteins.