BAY 87-2243 is a potent and selective hypoxia-inducible factor-1 (HIF-1) inhibitor.

PX-478 2HCl is an orally active, and selective hypoxia-inducible factor-1α (HIF-1α) inhibitor.

Alisertib is a selective Aurora A inhibitor.

Tozasertib is a pan-Aurora inhibitor.

Barasertib is a highly selective Aurora B inhibitor.

ZM 447439 is a selective and ATP-competitive inhibitor for Aurora A and Aurora B.

MLN8054 is a potent and selective inhibitor of Aurora A.

Danusertib is an Aurora kinase inhibitor for Aurora A/B/C.