ZM 306416 is a VEGFR (Flt and KDR) inhibitor.

SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.

Taxifolin, type I inhibitor for VEGFR-2 kinase, is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.

Canertinib is a pan-erbB tyrosine kinase inhibitor.

WZ4002 is a novel, mutant-selective EGFR inhibitor.

AC480 (BMS-599626) is a selective and efficacious inhibitor of HER1 and HER2.

Rociletinib is an orally available small molecule, irreversible inhibitor of epidermal growth factor receptor (EGFR) with potential antineoplastic activity.