BTB06584 is an IF1-dependent, selective inhibitor of the mitochondrial F1 Fo-ATPase.

Verdinexor (KPT-335) is an orally bioavailable, selective XPO1/CRM1 inhibitor.  

Bay K 8644 is a potent, selective activator of L-type Ca₂₊ channel with IC50 of 17.3 nM.

O4I1 is a potent Oct3/4 inducer.  

O4I2 is a potent Oct3/4 inducer, which is suitable for iPSC generation.  

SKF96365, originally identified as a blocker of receptor-mediated calcium entry, is widely used diagnostically, as a blocker of transient receptor potential canonical type (TRPC) channels.

Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM in CHrB30 cell line, reverses drug resistance in MDR cell Lines.

Optovin is a reversible photoactivated TRPA1 activator.