Udenafil(乌地那非) is a benzenesulfonamide derivative with vasodilatory activity.

Troglitazone(曲格列酮) is an orally-active thiazolidinedione with antidiabetic and hepatotoxic properties and potential antineoplastic activity.

Rosiglitazone(罗格列酮) is an orally-active thiazolidinedione with antidiabetic properties and potential antineoplastic activity.

IDO-IN-1 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor with an IC50 of 59 nM.

Disulfiram (二硫化四乙基秋兰姆) is a specific inhibitor of aldehyde-dehydrogenase (ALDH1), used for the treatment of chronic alcoholism by producing an acute sensitivity to alcohol.

Clofazimine (氯苯吩嗪) is a rhimophenazine dye, originally developed for the treatment of tuberculosis, it has both antimicrobial and antiinflammatory activity, postulated mechanisms of action include intercalation of clofazimine with bacterial DNA and increasing levels of cellular phospholipase A2.

Pioglitazone (匹格列酮) is a selective peroxisome proliferator-activated receptor-gamma (PPARγ) agonist, used to treat diabetes; A weak activator for full-length hPPARα, but not full-length hPPARδ.

Tioxolone (噻克索酮) is a metalloenzyme carbonic anhydrase I inhibitor with a Ki of 91 nM.