Doxazosin(甲磺酸多沙唑嗪), a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia.

Etodolac(依托度酸) is a nonsteroidal anti-inflammatory drug (NSAID) and a COX inhibitor, used for the treatment of inflammation and pain.

Felbamate(非氨酯) is an anticonvulsant drug used in the treatment of epilepsy NMDAR antagonist.

Flumazenil(氟马西尼) is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.

Fluvoxamine Maleate(马来酸氟伏沙明) is a selective serotonin (5-HT) reuptake inhibitor (SSRI), used in the treatment of obsessive-compulsive disorder.

Galanthamine(氢溴酸加兰他敏) is an AChE inhibitor with IC50 of 0.35 μM, exhibits 50-fold selectivity against butyryl-cholinesterase.

Loratadine(氯雷他定) is a histamine H1 receptor antagonist, used to treat allergies. Also acts as a selective inhibitor of B(0)AT2 with IC50 of 4 μM.

Mianserin(盐酸米安色林) is an potent antagonist of H1 histamine receptor and 5-HT serotonin receptors, used for the treatment of depression.