LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.  

KN-62 is a potent and specific inhibitor of Ca₂₊/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.9 μM also a non-competitive antagonist of the purinergic receptor P2RX7 (IC50 = 15 nM). It is selective for CaMKII relative to PKA, PKC and MLCK, but inhibits CaMKI and CaMKIV equally well, The Ki value of KN-62 for CaMK V is 0.8 μM.

KN-93 Phosphate is a potent and specific inhibitor of Ca₂₊/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.37 μM, no remarkable inhibitory effects on APK, PKC, MLCK or Ca₂₊-PDE activities.

NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.

L-685,458 is a specific and potent inhibitor of A beta PP gamma-secretase activity with Ki of 17 nM.  

A-438079 HCl is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9.  

SKF38393 HCl is a selective dopamine D1/D5 receptor agonist.  

PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents the severity of pulmonary arterial hypertension in the MCT rat model.