An inhibitor of DNA topoisomerase II

Cefotiam Hexetil Hydrochloride is a semi-synthetic cephalosporin antibiotic, and an antibacterial. the compound has broad spectrum activity against gram-positive and -negative bactera.

A Cox-2, iNOS, NOS II, and PGE2 inhibitor

A useful fluorochrome for histology, FRET and mitochondrial probe

Dexrazoxane(右雷佐生) is an anticancer drug able to block mitosis and to arrest dividing cells. It is an iron chelator and provides cardioprotection against anthracycline toxicity.

Clodronate(氯屈膦酸二钠四水合物) is a non-nitrogenous bisphosphonate that can bind to bone to reduce the bone resorption. It is used as an anti-osteoporotic drug for the prevention of osteoporosis in post-menopausal women and men.

A muscarinic receptor antagonist, specifically an H1 histamine receptor antagonist. This compound is a muscle relaxant. Orphenadrine has also been reported to inhibit the noradrenergic transporter and to block the NMDA receptor ion channel.

Hydroxyhexamide(乙酸己脲) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agents.