Verteporfin(维替泊芬) is a small molecule that inhibits TEAD–YAP association and YAP-induced liver overgrowth.

Plinabulin is an orally active diketopiperazine derivative with potential antineoplastic activity.

Degrasyn is a selective deubiquitinase (DUB: USP5, UCH-L1, USP9x, USP14, and UCH37) inhibitor.

Bafetinib (巴非替尼) is a potent and selective dual Bcr-Abl/Lyn inhibitor.

TAE684 is a potent and selective ALK inhibitor.

Fostamatinib disodium(福美司坦), a prodrug of the active metabolite R406, is a Syk inhibitor.

R406 (free base) is a potent Syk inhibitor.

Piceatannol, a natural stilbene, is a selective Syk inhibitor.