Molidustat (BAY 85-3934) is a potent hypoxia-inducible factor prolyl hydroxylase (HIF-PH) inhibitor.

PD-166866 is a selective inhibitor of FGFR1.

LW6 is a hypoxia-inducible factor 1(HIF) inhibitor.

IOX2 is a potent inhibitor of HIF-1α prolyl hydroxylase-2 (PHD2).

LFM-A13 is a specific Bruton's tyrosine kinase (BTK) inhibitor (IC50 = 2.5 μM).

PD173074 is a potent FGFR1 inhibitor.

Lorlatinib(劳拉替尼) is a potent, dual ALK/ROS1 inhibitor.

Vadimezan(2,5-己酮可可碱) is a vascular disrupting agents (VDA) and competitive inhibitor of DT-diaphorase.