Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor.

PF-562271 is a potent, ATP-competitive, reversible inhibitor of FAK.

PF-573228 is an ATP-competitive inhibitor of FAK.

PF-562271 HCl is the hydrochloride salt of PF-562271, which is a potent, ATP-competitive, reversible inhibitor of FAK.

PND-1186 is a reversible and selective FAK inhibitor.

CGI1746 is a potent and highly selective small-molecule inhibitor of the Btk.

ENMD-2076 has selective activity against Aurora A and Flt3 with IC50 of 14 nM and 1.86 nM, 25-fold selective for Aurora A than over Aurora B and less potent to VEGFR2/KDR and VEGFR3, FGFR1 and FGFR2 and PDGFRα.

Tamoxifen(他莫昔芬) is an antagonist of the estrogen receptor in breast tissue.