Memantine HCl(盐酸美金刚) is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively.
Cyproheptadine HCl(盐酸赛庚啶) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Lornoxicam(氯诺昔康) is a non-steroidal COX-1/COX-2 inhibitor, used as an anti-inflammatory drug to treat pain, osteoarthritis, and rheumatoid arthritis.
Orphenadrine Citrate(枸酸芬那君) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.
Terazosin HCl(盐酸特拉唑嗪二水合物) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
Famotidine(法莫替丁) is a histamine H2–receptor antagonist with IC50 of 0.6 mM, commonly used to treat heartburn, GERD, ulcers, and other digestive conditions.
Trimebutine(曲美布汀) is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain.
Ivabradine HCl(盐酸伊伐布雷定) a new If inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent.